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riluzole <chemical> A glutamate antagonist that has reported anticonvulsant activity. It has been shown to prolong the survival of patients with amyotrophic lateral sclerosis and has been approved in the united states to treat patients with als.
Pharmacological action: anaesthetics, anticonvulsants, excitatory amino acid antagonists, neuroprotective agents.
(12 Dec 1998)
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  • Riluzole - »õâ A glutamate antagonist (RECEPTORS, GLUTAMATE) used as an anticonvulsant (ANTICONVULSANTS) and to prolong the survival of patients with AMYOTROPHIC LATERAL SCLEROSIS.
    Synonyms : 2-Amino-6-trifluoromethoxybenzothiazole, PK-26124, RP-54274, Rilutek, 2 Amino 6 trifluoromethoxybenzothiazole
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Aventis
E02830081 Riluzole
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E06400461 Riluzole
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riluzole (ril
Ãâó: www.mercksource.com/pp/us/cns/cns_hl_dorlands.jspz...
riluzole Riluzole is a drug used to treat amyotrophic lateral sclerosis. It delays the onset of ventilator-dependence in selected patients and may increase survival by approximately two months. A Cochrane Library review states a 9% gain in the probability of surviving one year. In secondary analyses of survival at separate time points, there was a significant survival advantage with Riluzole 100 mg at six, nine, 12 and 15 months, but not at three or 18 months. ...
Ãâó: en.wikipedia.org/wiki/Riluzole
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