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technetium tc 99m exametazime <chemical> A gamma-emitting radionuclide imaging agent used in the evaluation of regional cerebral blood flow and in non-invasive dynamic biodistribution studies and myocardial imaging. It has also been used to label leukocytes in the investigation of inflammatory bowel diseases.
Pharmacological action: radiopharmaceuticals.
(12 Dec 1998)
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exametazime HMPAO; hexamethylpropyleneamine oxime, a neutral lipophilic compound that traverses the blood-brain barrier and localizes in the brain; complexed with technetium 99m it is used for imaging of cerebral regional blood flow in the detection of altered regional perfusion in stroke, identification of Alzheimer's disease, evaluation of epilepsy, and diagnosis of brain death. The same complex can also be used to label autologous leukocytes for diagnostic studies of intra-abdominal inflammatory lesions and bowel disease. See table at technetium.
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