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baclofen <chemical> A gaba derivative that is a specific agonist at gaba-b receptors (receptors, gaba-b). It is used in the treatment of spasticity, especially that due to spinal cord damage. Its therapeutic effects result from actions at spinal and supraspinal sites, generally the reduction of excitatory transmission.
Pharmacological action: gaba agonists, muscle relaxants, central.
Chemical name: Benzenepropanoic acid, beta-(aminomethyl)-4-chloro-
(12 Dec 1998)
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  • Baclofen - »õâ A GAMMA-AMINOBUTYRIC ACID derivative that is a specific agonist at GABA-B receptors (RECEPTORS, GABA-B). It is used in the treatment of spasticity, especially that due to spinal cord damage. Its therapeutic effects result from actions at spinal and supraspinal sites, generally the reduction of excitatory transmission.
    Synonyms : ASTA Medica Brand of Baclofen, Alphapharm Brand of Baclofen, Apo-Baclofen, Apotex Brand of Baclofen, Ashbourne Brand of Baclofen, Athena Brand of Baclofen, Atrofen, Ba-34, 647, Ba-34647, Baclofen AWD, Baclofene-Irex, Baclospas, CIBA-34, 647-BA, Clofen, Gen-Baclofen
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baclofen A mainstay of antispastic drug therapy, baclofen is a GABA agonist that stimulates the GABAB autoreceptor. When stimulated, this autoreceptor inhibits muscle activity. In experimental systems, baclofen inhibits the release of noradrenaline, and acetylcholine from peripheral nerve endings, and acetylcholine, noradrenaline, dopamine, serotonin, and glutamate from CNS neurons.
Ãâó: www.dbs-stn.org/glossary.asp
baclofen A medication used to reduce spasticity.
Ãâó: cerebralpalsylawyers.homestead.com/cerebral_palsy_...
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